Testifenon


Testifenon, also known as testiphenon, testiphenone, chlorphenacyl dihydrotestosterone ester, or dihydrotestosterone 17β-acetate, is a synthetic anabolic–androgenic steroid and a cytostatic antineoplastic agent that was never marketed. It is an androgen esterspecifically, a chlorphenacyl nitrogen mustard ester of dihydrotestosterone – and acts as a prodrug of these two components in the body. The drug was developed in Russia as a tissue-selective cytostatic drug for the treatment of various cancers occurring in androgen receptor-expressing tissues that would have reduced side effects and toxicity relative to other chemotherapy drugs.